1094-2009 Publicatins

1094-2009 Publicatins

 

1. “Synthesis of Pyrido[2,3.4-kl]Acridines. A Building Block for synthesis of pyridoacridine alkaloids”, Gellerman G., Rudi A., Kashman Y., Tetrahedron Letters, 33, 5577-5580, 1992.

2. “Biomimetic Synthesis of Pyrido[2,3.4-kl]Acridines”, Gellerman G., Rudi A., Kashman Y., Tetrahedron Letters, 34, 1823-1826, 1993.

3. “A Two Step Biomimetic Total Synthesis of Eilatin”, Gellerman G., Babad M., Kashman Y., Tetrahedron Letters, 34, 1827-1830, 1993.

4. “Biomimetic Synthesis of Ascididemin and Derivatives”, Gellerman G., Rudi A., Kashman Y., Synthesis, 3, 239-241, 1994.

5. “The Biomimetic Synthesis of Marine Alkaloide releated Pyrido- and Pyrrolo[2,3.4-kl]Acridines”, Gellerman G., Rudi A., Kashman Y., Tetrahedron, 50, 12959-12972, 1994.

6. “Potent Antileukemic Effect of some Pyridoacredine Alkaloides”, Einat M., Elishner M., Nagler A., Fabian I., Gellerman G., Rudi A., Kashman Y., Clinical Canser Research, 1, 823-829, 1995.

7. ”A Backbone-Cyclic, receptor 5 selective somatostatin analogue: synthesis, bioactivity, and NMR conformational analysis” Gilon C., Huenges M., Matha B., Gellerman G., Kessler H., Journal of Medicinal Chemistry, 41, 919-929, 1998.

8. “Facil Synthesis of Orthogonally Protected Amino Acid Building Blocks for Combinatorial and Backbone Cyclic Peptide Chemistry”, Gellerman G., Elgavi A., Kramer M., Journal of Peptide Research, 57, 277-290, 2001.

9. “Human Somatostatin Receptor Specificity of Backbone-Cyclic Analogues Containing Novel Sulfur Building Units”, Gazal S., Gellerman G., Ziv O., Karpov O., Litman P., Bracha M., Afargan M., Gilon C., Journal of Medicinal Chemistry, 45, 1665-1671, 2002.

10. ”Synthesis of Novel Protected Na(w-thioalkyl) Amino Acid Building Units and their Incorporation in Backbone Cyclic Disulfide and Thioetheric Bridged Peptides” Gazal S., Gellerman G., Glukhov E., Gilon C., Journal of Peptide Research, 58, 527-539. 2001.

11. “Bioactive Somatostatin Analog Without a type II’ beta-turn: Synthesis and Conformational Analysis in Solution”. Jiang S., Gazal S., Gellerman G., Ziv O., Karpov O., Litman P., Bracha M., Afargan M., Gilon C., Goodman M. A., Journal of Peptide Science, 7, 521-528, 2001.

12. “Novel Gly Building Units for Backbone Cyclization: Synthesis and Incorporation Into Model Peptides”. Gazal S, Gellerman G, Gilon C., Peptides, 24, 1847-1852, 2003.

13. “Long-Acting SST Analog with Endocrine Selectivity: Potent suppression of Growth Hormone but not of Insulin”. Afargan M., Tiensuu E., Gellerman G., Oberg K., Endocrinology, 142, 477-486, 2001.

14. “Toward a PKB Inhibitor: Modification of a Selective PKA Inhibitor by Rational Design”, Reuveni H., Livnah N., Geiger T., Klein S., Ohne O., Cohen I., Benhar M., Gellerman G., Levitzki A., Biochemistry, 41, 10304-10314, 2002.

15. “A facile two-step synthesis of Novel ring-A double substituted tryptophan building blocks for combinatorial chemistry”, Gorohovsky S., Meir S., Shkoulev V., Byk G., Gellerman G., Synlett, 10, 1411-1414, 2003.

16. “Dilactams. Synthesis of nonsymmetrical dibenzodiazocinediones”, Hassner A., Sun B., Gellerman G., Meir S., Tetrahedron Letters, 45, 1377-1379, 2004.

17. “New application of DPPA reagent: one pot transformation of quinolin-4-one and pyridin-4-one derivatives into 4-azido and 4-amino counterparts.” Aizikovich A., Kuznetsov V., Gorohovsky S., Levy A., Meir S., Byk G., Gellerman G., Tetrahedron Letters, 45, 4241-4243, 2004.

18. “Approaches for introducing high molecular diversity in scaffolds: Fast Parallel Synthesis of Highly Substituted 1H-quinolin-4-one Libraries” Kuznetsov V., Gorohovsky S., Levy A., Meir S., Shkoulev V., Menashe N., Greenwald M., Aizikovich A., Ofer D., Byk G., Gellerman G., Molecular Diversity, 8, 437-448, 2004.

19. “Reductive Nitrosation of Peptides Ligated to High Valent Metal Cations”, Shamir D., Zilbermann I., Maimon E., Gellerman G., Cohen H., Meyerstein D., Eur. Jour. Inorg. Chem., 32, 5029-5031, 2007.

20. “Facile Synthesis of Orthogonally Protected Optically Pure Keto- and Diketopiperazine Building Blocks for Combinatorial Chemistry”, Gellerman G., Hazan E., Albeck A., Shatzmiler S., Intern. Jour. Pep. Res. Ther, 14, 183-192, 2008.

21. “Synthesis of Orthogonally Protected Optically Pure Ketopiperazine, Diketopiperazine, Ketodiazepane and 3-Aminopyrrolidone Building Blocks for Peptidomimetic Combinatorial Chemistry”, Gellerman G., Hazan E., Albeck A., Shatzmiler S., Tetrahedron, 65, 1389–1396, 2009.

22. “Synthesis of chiral heteronucleotide ONA sequences by a Fmoc/Boc-based
submonomeric strategy” Amir A., Hetsron A., Shatzmiller S., Gellerman G., Intern. Jour. Pep. Res. Ther., 15, 241-246, 2009.

23. “Synthesis and Antifungal Activity of β-Trifluroalkyl Aminovinyl Ketone Derivatives”, Gellerman G., Pariente N., Paz Z., Shneiderman A., Yarden O., Agric. Food Chem., 57, 8303-8307, 2009.